InChIKey	VHYCDWMUTMEGQY-UHFFFAOYSA-N
Compound Name	Bisoprolol
Canonical SMILES	CC(C)NCC(O)COc1ccc(COCCOC(C)C)cc1
Clinical Status	Data-mined Candidate
Targets (Human+Pathogen)	2
Pfam Stratification	Homologous
Avg pChEMBL	7.25
Source	BindingDB;ChEMBL

DrugBank ID	DB00612
Drug Name	Bisoprolol
CAS Number	66722-44-9
Groups	approved investigational
ATC Codes	C07FX04 C07BB07 C07AB07 C09BX05 C09BX02 C09BX04 C09BX06 C07FB07
Description	Bisoprolol is a cardioselective β1-adrenergic blocking agent used to treat high blood pressure.[A180472,L7219] It is considered a potent drug with a long-half life that can be used once daily to reduce the need for multiple doses of antihypertensive drugs.[A180472] Bisoprolol is generally well toler...

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Categories: Adrenergic Agents Adrenergic Antagonists Adrenergic beta-1 Receptor Antagonists Adrenergic beta-Antagonists Agents causing hyperkalemia Alcohols Amines Amino Alcohols Antiarrhythmic agents Antihypertensive Agents Antihypertensive Agents Indicated for Hypertension Autonomic Agents Beta Blocking Agents and Thiazides Beta Blocking Agents, Selective Beta Blocking Agents, Selective, and Thiazides Beta blocking agents and calcium channel blockers Beta-Blockers (Beta1 Selective) Bradycardia-Causing Agents Cardiovascular Agents Cytochrome P-450 CYP3A Substrates Cytochrome P-450 CYP3A4 Substrates Cytochrome P-450 Substrates Drugs that are Mainly Renally Excreted Hypotensive Agents Neurotransmitter Agents P-glycoprotein inhibitors P-glycoprotein substrates Peripheral Nervous System Agents Phenoxypropanolamines Propanolamines Propanols Sympatholytics

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Cross-references: BindingDB: 25751 ChEBI: 3127 CHEMBL645 ChemSpider: 2312 Drugs Product Database (DPD): 1218 C06852 D02342 PharmGKB: PA448641 PubChem:2405 PubChem:46508844 RxCUI: 19484 Therapeutic Targets Database: DAP000483 Wikipedia: Bisoprolol