Molecule Details
InChIKeyVHJQAYMEVPBDIB-UHFFFAOYSA-N
Compound Name2-(4-(1H-imidazol-1-yl)phenoxy)-N-([1,1'-biphenyl]-4-yl)acetamide
Canonical SMILESO=C(COc1ccc(-n2ccnc2)cc1)Nc1ccc(-c2ccccc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H237 PORCN Homo sapiens Human PF03062 7.8 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 7.7 IC50 ChEMBL;BindingDB
P10635 CYP2D6 Homo sapiens Human PF00067 7.0 IC50 ChEMBL;BindingDB