Molecule Details
InChIKeyVGWGODQLJSCOSQ-UHFFFAOYSA-N
Compound Name2-Methyl-4-[4-(4-sulfamoylanilino)phthalazin-1-yl]benzenesulfonamide
Canonical SMILESCc1cc(-c2nnc(Nc3ccc(S(N)(=O)=O)cc3)c3ccccc23)ccc1S(N)(=O)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.71
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16790 CA9 Homo sapiens Human PF00194 8.5 IC50 ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.6 IC50 ChEMBL;BindingDB
P00915 CA1 Homo sapiens Human PF00194 7.1 IC50 ChEMBL;BindingDB