Molecule Details
InChIKeyVGVIWBCNXYVLQY-UHFFFAOYSA-N
Compound NameTert-Butyl 6-{[2-Chloro-4-(Dimethylcarbamoyl)phenyl]amino}-2-(1,3-Oxazol-5-Yl)-1h-Pyrrolo[3,2-C]pyridine-1-Carboxylate
Canonical SMILESCN(C)C(=O)c1ccc(Nc2cc3c(cn2)cc(-c2cnco2)n3C(=O)OC(C)(C)C)c(Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P20248 CCNA2 Homo sapiens Human PF02984 PF00134 PF16500 6.8 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB