Molecule Details
InChIKeyVFRGUPCPOYDATL-UHFFFAOYSA-N
Compound Name1-[4-[6-(1H-indazol-5-ylamino)pyrimidin-4-yl]oxynaphthalen-1-yl]-3-[1-(4-methoxyphenyl)-3-propan-2-ylpyrazol-5-yl]urea
Canonical SMILESCOc1ccc(-n2nc(C(C)C)cc2NC(=O)Nc2ccc(Oc3cc(Nc4ccc5[nH]ncc5c4)ncn3)c3ccccc23)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.0 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.4 IC50 ChEMBL;BindingDB