Molecule Details
InChIKeyVFQLHOJNCNGPIK-SANMLTNESA-N
Compound Name6-Methyl-4''-trifluoromethyl-biphenyl-2-carboxylic acid {2-[(pyridin-2-ylmethyl)-amino]-indan-5-yl}-amide
Canonical SMILESCc1cccc(C(=O)Nc2ccc3c(c2)C[C@@H](NCc2ccccn2)C3)c1-c1ccc(C(F)(F)F)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.56
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P04114 APOB Homo sapiens Human PF12491 PF06448 PF09172 PF01347 8.8 IC50 ChEMBL;BindingDB
P55157 MTTP Homo sapiens Human PF19444 PF01347 7.0 IC50 ChEMBL;BindingDB
Q99835 SMO Homo sapiens Human PF01534 PF01392 6.9 IC50 ChEMBL;BindingDB