Molecule Details
InChIKeyVFKIKYZNUCGJGD-UHFFFAOYSA-N
Compound Name1-(5',11'-Dihydrospiro[cyclopentane-1,10'-dibenzo[a,d]cyclohepten]-3-yl)-1,2,3,6-tetrahydro-4-pyridinecarboxylic acid
Canonical SMILESO=C(O)C1=CCN(C2CCC3(Cc4ccccc4Cc4ccccc43)C2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.07
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35367 HRH1 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.1 Ki ChEMBL
P28335 HTR2C Homo sapiens Human PF00001 6.7 Ki ChEMBL