Molecule Details
InChIKeyVFIZBHJTOHUOEK-UHFFFAOYSA-N
Compound NameS-Ethylisothiourea
Canonical SMILESCCSC(=N)N
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB02234
Drug NameS-Ethylisothiourea
CAS Number2986-20-1
Groups investigational
ATC Codes nan
DescriptionS-Ethylisothiourea is a nitric oxide synthase inhibitor.

Categories: Amides Cardiovascular Agents Central Nervous System Agents Central Nervous System Depressants Enzyme Inhibitors Hypnotics and Sedatives Nitric Oxide Synthase, antagonists & inhibitors Sulfur Compounds Thiourea Vasoconstrictor Agents
Cross-references: BindingDB: 50055281 CHEMBL321691 ChemSpider: 4955 PDB: ITU PubChem:5139 PubChem:46508006 ZINC: ZINC000003806245
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29475 NOS1 Homo sapiens Human PF00667 PF00258 PF00175 PF02898 PF00595 7.5 Ki ChEMBL;BindingDB
P29474 NOS3 Homo sapiens Human PF00667 PF00258 PF00175 PF02898 7.4 Ki ChEMBL
P35228 NOS2 Homo sapiens Human PF00667 PF00258 PF00175 PF02898 6.8 IC50 ChEMBL;BindingDB
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P0A094 P0A094 Nitric oxide synthase oxygenase binder targets
P29474 NOS3 Nitric oxide synthase 3 inhibitor targets
P35228 NOS2 Nitric oxide synthase, inducible inhibitor targets