Molecule Details
InChIKeyVFESYYJORSLMBC-UHFFFAOYSA-N
Canonical SMILESCc1cnc(-c2ccnc(C(C)(C)CO)n2)c(F)c1-n1c(C)cc(OCc2ncc(F)cc2F)c(Cl)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.75
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8IW41 MAPKAPK5 Homo sapiens Human PF00069 9.0 IC50 BindingDB
P49137 MAPKAPK2 Homo sapiens Human PF00069 6.5 IC50 BindingDB