Molecule Details
InChIKeyVEWFKNUERSAOIS-UHFFFAOYSA-N
Compound Name2-Amino-5-(3-aminophenyl)-3-(oxolan-2-ylmethyl)-7-phenylquinazolin-4-one
Canonical SMILESNc1cccc(-c2cc(-c3ccccc3)cc3nc(N)n(CC4CCCO4)c(=O)c23)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.03
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P46925 PMII Plasmodium falciparum (isolate HB3) Pathogen PF00026 6.1 IC50 ChEMBL;BindingDB
Q17SB2 Plasmodium falciparum Pathogen PF00026 6.0 IC50 ChEMBL
Q8IM16 PMIV Plasmodium falciparum (isolate 3D7) Pathogen PF00026 6.0 IC50 BindingDB