Molecule Details
InChIKeyVETBKPDTHQZBKH-UHFFFAOYSA-N
Compound Name1-(4-(3-(Trifluoromethyl)phenethyl)benzyl)azetidine-3-carboxylic acid
Canonical SMILESO=C(O)C1CN(Cc2ccc(CCc3cccc(C(F)(F)F)c3)cc2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H228 S1PR5 Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P21453 S1PR1 Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
P34947 GRK5 Homo sapiens Human PF00069 PF00615 6.1 Ki ChEMBL