Molecule Details
InChIKeyVELBXKDYGYBFSC-UHFFFAOYSA-N
Compound Name4-(1-isopropyl-2-methyl-1H-imidazol-5-yl)-N-(4-((tetrahydrofuran-2-yl)methylsulfonyl)phenyl)pyrimidin-2-amine
Canonical SMILESCc1ncc(-c2ccnc(Nc3ccc([S@SP3](=O)(=O)CC4CCCO4)cc3)n2)n1C(C)C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.89
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.9 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.9 pIC50 TTD_MultiTarget