Molecule Details
InChIKeyVDXFKYHWRXWVOF-IBGZPJMESA-N
Compound NameN-[3-[(6R)-4-amino-2-cyano-6-methyl-7H-pyrazolo[1,5-a]pyrazin-6-yl]-4-fluorophenyl]-2-methyl-1,3-oxazole-4-carboxamide
Canonical SMILESCc1nc(C(=O)Nc2ccc(F)c([C@]3(C)Cn4nc(C#N)cc4C(N)=N3)c2)co1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5Z0 BACE2 Homo sapiens Human PF00026 9.5 Ki ChEMBL;BindingDB
P56817 BACE1 Homo sapiens Human PF00026 8.8 IC50 ChEMBL;BindingDB
P05067 APP Homo sapiens Human PF10515 PF12924 PF12925 PF02177 PF03494 PF00014 8.3 IC50 ChEMBL;BindingDB