Molecule Details
InChIKeyVDNQILFFXZGSAK-UHFFFAOYSA-N
Compound Name4-((2-methylquinolin-4-yl)methoxy)-N-((2,4,6-trioxo-5-(4-pivaloylpiperazin-1-yl)-hexahydropyrimidin-5-yl)methyl)benzamide
Canonical SMILESCc1cc(COc2ccc(C(=O)NCC3(N4CCN(C(=O)C(C)(C)C)CC4)C(=O)NC(=O)NC3=O)cc2)c2ccccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.7 Ki ChEMBL;BindingDB
P39900 MMP12 Homo sapiens Human PF00045 PF00413 PF01471 7.3 Ki ChEMBL;BindingDB