Molecule Details
InChIKeyVCZRYZZCLOMGOV-UHFFFAOYSA-N
Compound NameN-(6-piperazin-1-yl-3-pyridinyl)-4-(2-pyrrolidin-1-ylquinazolin-6-yl)pyrimidin-2-amine
Canonical SMILESc1cc(-c2ccc3nc(N4CCCC4)ncc3c2)nc(Nc2ccc(N3CCNCC3)nc2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL7.56
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86YV6 MYLK4 Homo sapiens Human PF00069 8.7 IC50 ChEMBL
Q9UEE5 STK17A Homo sapiens Human PF00069 7.8 IC50 ChEMBL
Q9HAZ1 CLK4 Homo sapiens Human PF00069 6.9 IC50 ChEMBL
Q9UHD2 TBK1 Homo sapiens Human PF00069 PF18394 PF18396 6.9 IC50 ChEMBL