Molecule Details
InChIKeyVCASZZUAVHWYHQ-UHFFFAOYSA-N
Compound Name4-[(5-Formamidocyclohexa-2,4-dien-1-yl)methylamino]quinazoline-8-carboxamide
Canonical SMILESNC(=O)c1cccc2c(NCC3C=CC=C(NC=O)C3)ncnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.64
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 9.3 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 9.2 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.4 IC50 ChEMBL;BindingDB