Molecule Details
InChIKeyVCADIWSEVTZZOR-UHFFFAOYSA-N
Compound Name6-chloro-N-(furan-3-ylmethyl)-2-(4-methylpiperazin-1-yl)quinazolin-4-amine
Canonical SMILESCN1CCN(c2nc(NCc3ccoc3)c3cc(Cl)ccc3n2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P46098 HTR3A Homo sapiens Human PF02931 PF02932 8.6 Ki ChEMBL;BindingDB
Q9H3N8 HRH4 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P35367 HRH1 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB