Molecule Details
InChIKeyVBQONCXEWJGAOC-UHFFFAOYSA-N
Compound Name4-[(5-methylthieno[2,3-d]pyrimidin-4-yl)amino]-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamide
Canonical SMILESCc1csc2ncnc(Nc3c[nH]nc3C(=O)Nc3ccc(CN4CCOCC4)cc3)c12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P78396 CCNA1 Homo sapiens Human PF02984 PF00134 PF16500 9.0 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
P36888 FLT3 Homo sapiens Human PF00047 PF07714 8.9 IC50 ChEMBL;BindingDB