Molecule Details
InChIKeyVBBBMBNPLKHHEO-UHFFFAOYSA-N
Canonical SMILESCCOc1nc(Cl)ccc1C1(N2CCN(c3ccncc3)CC2)C(=O)N(S(=O)(=O)c2ccc(OC)cn2)c2ccc(C#N)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P47901 AVPR1B Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 7.0 IC50 ChEMBL;BindingDB