Molecule Details
InChIKeyVAWVZAYWTUKBNV-UHFFFAOYSA-N
Compound NameN-{4-[3-amino-1-(2-methoxyethyl)-1H-indazol-4-yl]phenyl}-N''-(2-fluoro-5-methylphenyl)urea
Canonical SMILESCOCCn1nc(N)c2c(-c3ccc(NC(=O)Nc4cc(C)ccc4F)cc3)cccc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.32
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.3 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.3 pIC50 TTD_MultiTarget