Molecule Details
InChIKeyVAUKHARIAMDAGF-UHFFFAOYSA-N
Compound NameN-[4-[(Dimethylamino)sulfonyl]phenyl]-4-(hydroxydiphenylmethyl)-1-piperidinecarbothioamide
Canonical SMILESCN(C)S(=O)(=O)c1ccc(NC(=S)N2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49146 NPY2R Homo sapiens Human PF00001 7.7 IC50 ChEMBL;BindingDB
Q5BJF2 TMEM97 Homo sapiens Human PF05241 6.6 Ki ChEMBL
P30536 TSPO Homo sapiens Human PF03073 6.0 Ki ChEMBL