Molecule Details
InChIKeyVAKWGLDYQAWDPS-UHFFFAOYSA-N
Compound Nametert-butyl 4-(4-(5-methyl-1H-pyrazol-3-ylamino)quinazolin-2-ylthio)phenylcarbamate
Canonical SMILESCc1cc(Nc2nc(Sc3ccc(NC(=O)OC(C)(C)C)cc3)nc3ccccc23)n[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.57
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.1 Ki ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 8.1 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.6 Ki ChEMBL;BindingDB