Molecule Details
InChIKeyUZWNDXWGPCUGGI-HDICACEKSA-N
Compound Name4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-{3-[(3R,5S)-3,4,5-trimethylpiperazin-1-yl]propoxy}quinoline-3-carbonitrile
Canonical SMILESCOc1cc(Nc2c(C#N)cnc3cc(OCCCN4C[C@@H](C)N(C)[C@@H](C)C4)c(OC)cc23)c(Cl)cc1Cl
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.85
SourceBindingDB;TTD_MultiTarget
2D Structure
2D structure
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.8 IC50 BindingDB
P00519 ABL1 Homo sapiens Human PF08919 PF07714 PF00017 PF00018 Clinical TTD_MultiTarget TTD_MultiTarget