Molecule Details
InChIKeyUZWFLOSUVZITCB-UHFFFAOYSA-N
Compound NameN-(3-fluorophenyl)-2-(2-(7-(3-(2-hydroxyethylamino)propoxy)-6-methoxyquinazolin-4-ylamino)thiazol-5-yl)acetamide
Canonical SMILESCOc1cc2c(Nc3ncc(CC(=O)Nc4cccc(F)c4)s3)ncnc2cc1OCCCNCCO
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.3
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 8.3 pIC50 TTD_MultiTarget