Molecule Details
InChIKeyUZSMYCXKQUZNLV-UHFFFAOYSA-N
Compound Name4-(1-Benzyl-piperidin-4-yl)-6-(4-chloro-phenyl)-pyrimidin-2-ylamine
Canonical SMILESNc1nc(-c2ccc(Cl)cc2)cc(C2CCN(Cc3ccccc3)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 8.1 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB