Molecule Details
InChIKeyUZRQKIJPXLTOGR-UHFFFAOYSA-N
Compound Name[4-[(5-Sulfamoyl-1,3,4-thiadiazol-2-yl)sulfamoyl]anilino] morpholine-4-carbodithioate
Canonical SMILESNS(=O)(=O)c1nnc(NS(=O)(=O)c2ccc(NSC(=S)N3CCOCC3)cc2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.67
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 8.8 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.8 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 8.3 Ki ChEMBL;BindingDB