Molecule Details
InChIKeyUYRUHHLEYUGTMC-UHFFFAOYSA-N
Compound Name7-[(3-Bromophenyl)methyl]-1-methyl-5,6-dihydrotriazolo[1,5-d][1,4]benzodiazepine
Canonical SMILESCc1nnn2c1-c1ccccc1N(Cc1cccc(Br)c1)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.7 IC50 ChEMBL;BindingDB
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.7 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.1 IC50 ChEMBL;BindingDB