Molecule Details
InChIKeyUYQKRAKNSZLAGM-UHFFFAOYSA-N
Compound Name2-[3-(6-cyclopropylpyrazin-2-yl)-1H-indol-5-yl]-5-(1H-pyrazol-5-yl)-1,3,4-oxadiazole
Canonical SMILESc1cc(-c2nnc(-c3ccc4[nH]cc(-c5cncc(C6CC6)n5)c4c3)o2)[nH]n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB