Molecule Details
InChIKeyUYKNWWODISPUHU-UHFFFAOYSA-N
Canonical SMILESCN1CCN(CCCNc2ncnc3c2cnn3-c2ccc(OCCCc3sc(N4CCc5cccc(C(=O)Nc6nc7ccccc7s6)c5C4)nc3C(=O)O)cc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.68
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 10.5 Ki ChEMBL;BindingDB
P10415 BCL2 Homo sapiens Human PF00452 PF02180 6.8 Ki ChEMBL;BindingDB