Molecule Details
InChIKeyUYFVVRGISWEBNS-YRNVUSSQSA-N
Compound Name4-[(E)-3-(hydroxyamino)-3-oxoprop-1-enyl]-N-[4-methyl-3-[(5-pyridin-3-yl-1,3-thiazol-2-yl)amino]phenyl]benzamide
Canonical SMILESCc1ccc(NC(=O)c2ccc(/C=C/C(=O)NO)cc2)cc1Nc1ncc(-c2cccnc2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.2
SourceBindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 7.4 IC50 BindingDB
Q02161 RHD Homo sapiens Human PF00909 7.1 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 7.1 pIC50 TTD_MultiTarget