Molecule Details
InChIKeyUXZATHOFDZQOMY-UHFFFAOYSA-N
Compound Name3-(Cyclopropylamino)-5-(3-(trifluoromethyl)phenylamino)pyrimido(4,5-c)quinoline-8-carboxylic acid
Canonical SMILESO=C(O)c1ccc2c(c1)nc(Nc1cccc(C(F)(F)F)c1)c1nc(NC3CC3)ncc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Cross-Family
Avg pChEMBL8.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P68400 CSNK2A1 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P19784 CSNK2A2 Homo sapiens Human PF00069 8.0 IC50 ChEMBL
P67870 CSNK2B Homo sapiens Human PF01214 8.0 IC50 ChEMBL
Q8NEV1 CSNK2A3 Homo sapiens Human PF00069 8.0 IC50 ChEMBL