Molecule Details
InChIKeyUXROPHBUPUPWOI-BQZHBXIKSA-N
Compound Name(2S)-N-[(2S,3S)-3-hydroxy-5-[[(2S)-4-methyl-1-[[(2S)-1-[methyl-[(2R)-1-oxo-3-phenyl-1-(propan-2-ylamino)propan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopentan-2-yl]amino]-5-oxo-1-phenylpentan-2-yl]-2-[[(2S)-2-[[(2S)-2-hydroxypropanoyl]amino]-3-methylbutanoyl]-methylamino]pentanediamide
Canonical SMILESCC(C)C[C@H](NC(=O)C[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(N)=O)N(C)C(=O)[C@@H](NC(=O)[C@H](C)O)C(C)C)C(=O)N[C@@H](C)C(=O)N(C)[C@H](Cc1ccccc1)C(=O)NC(C)C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.89
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14091 CTSE Homo sapiens Human PF07966 PF00026 7.3 IC50 ChEMBL;BindingDB
P56817 BACE1 Homo sapiens Human PF00026 6.8 IC50 ChEMBL;BindingDB
P07339 CTSD Homo sapiens Human PF07966 PF00026 6.6 IC50 ChEMBL;BindingDB