Molecule Details
InChIKeyUXDZDQRAGSHUBW-UHFFFAOYSA-N
Compound Name2-Ethyl-1-(3-fluorophenyl)sulfonyl-4-piperazin-1-ylimidazo[4,5-c]pyridine
Canonical SMILESCCc1nc2c(N3CCNCC3)nccc2n1S(=O)(=O)c1cccc(F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.03
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50406 HTR6 Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB