Molecule Details
InChIKeyUWTMXZFDTBHJPH-UHFFFAOYSA-N
Compound Name8-[3-chloro-5-[3-(methylamino)-1H-indazol-6-yl]-4-pyridinyl]-2,8-diazaspiro[4.5]decan-1-one
Canonical SMILESCNc1n[nH]c2cc(-c3cncc(Cl)c3N3CCC4(CCNC4=O)CC3)ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49336 CDK8 Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
Q9BWU1 CDK19 Homo sapiens Human PF00069 8.5 IC50 ChEMBL
P24863 CCNC Homo sapiens Human PF16899 PF00134 8.5 IC50 ChEMBL