Molecule Details
InChIKeyUVJRFPDIIZDNQE-UHFFFAOYSA-N
Compound NameN-(azetidin-3-yl)-5-[3-(6-cyclopropylpyrazin-2-yl)-1H-indol-5-yl]-1,3,4-oxadiazol-2-amine
Canonical SMILESc1cc2[nH]cc(-c3cncc(C4CC4)n3)c2cc1-c1nnc(NC2CNC2)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.5 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 8.9 IC50 ChEMBL;BindingDB