Molecule Details
InChIKeyUUYUVYXSHUTRGO-UHFFFAOYSA-N
Compound Name5,7-Dichloro-4-(5-chloro-2-hydroxyphenyl)-3-hydroxy-2(1H)-quinolinone
Canonical SMILESO=c1[nH]c2cc(Cl)cc(Cl)c2c(-c2cc(Cl)ccc2O)c1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL6.25
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96KB5 PBK Homo sapiens Human PF00069 6.5 Ki ChEMBL
Q9HAZ1 CLK4 Homo sapiens Human PF00069 6.4 Ki ChEMBL
Q13627 DYRK1A Homo sapiens Human PF00069 6.1 Ki ChEMBL
P11309 PIM1 Homo sapiens Human PF00069 6.0 Ki ChEMBL