Molecule Details
InChIKeyUUQDXDINAPCENI-UHFFFAOYSA-N
Compound NameN-(7-(N-ethylacetamido)-4-methoxybenzo[d]thiazol-2-yl)-4-(piperidine-1-carbonyl)benzamide
Canonical SMILESCCN(C(C)=O)c1ccc(OC)c2nc(NC(=O)c3ccc(C(=O)N4CCCCC4)cc3)sc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 8.1 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB