Molecule Details
InChIKeyUUKCYLIDEZGIBS-IBGZPJMESA-N
Compound Name(S)-2-(1,1-dioxo-1lambda*6*-thiomorpholin-4-yl)-N-hydroxy-3-{methanesulfonyl-[4-(4-trifluoromethyl-phenoxy)-phenyl]-amino}-propionamide
Canonical SMILESCS(=O)(=O)N(C[C@@H](C(=O)NO)N1CCS(=O)(=O)CC1)c1ccc(Oc2ccc(C(F)(F)F)cc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.54
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.8 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.3 pIC50 TTD_MultiTarget