Molecule Details
InChIKeyUUISESFNPSRBFN-UHFFFAOYSA-N
Compound Name2-[(2-Bromo-4-methylphenyl)[6-({4-[3-(dimethylamino)-2-hydroxypropoxy]phenyl}amino)pyrimidin-4-yl]amino]acetonitrile
Canonical SMILESCc1ccc(N(CC#N)c2cc(Nc3ccc(OCC(O)CN(C)C)cc3)ncn2)c(Br)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.0
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget