Molecule Details
InChIKeyUTWLDWAFEKZNCC-UHFFFAOYSA-N
Canonical SMILESCOc1ccc(F)cc1-c1cc(C)ncc1C(=O)Nc1nnc(OC2CC3(CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)C2)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.73
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P09874 PARP1 Homo sapiens Human PF00533 PF21728 PF00644 PF02877 PF05406 PF00645 PF08063 8.3 IC50 ChEMBL
O75417 POLQ Homo sapiens Human PF00270 PF00476 PF25453 PF00271 PF20470 PF21099 7.1 IC50 ChEMBL