Molecule Details
InChIKeyUSPFJPDEADLGIG-HSZRJFAPSA-N
Compound Name(20S)-19,20,21,22-Tetrahydro-19-oxo-5H-18,20-ethano-12,14-etheno-6,10-metheno-18H-benz(D)imidazo(4,3-K)(1,6,9,12)oxatriaza-cyclooctadecosine-9-carbonitrile
Canonical SMILESN#Cc1ccc2cc1Oc1ccc3cccc(c3c1)N1CC[C@@H](NCc3cncn3C2)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.8
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB08674
Drug Name(20S)-19,20,21,22-TETRAHYDRO-19-OXO-5H-18,20-ETHANO-12,14-ETHENO-6,10-METHENO-18H-BENZ[D]IMIDAZO[4,3-K][1,6,9,12]OXATRIAZA-CYCLOOCTADECOSINE-9-CARBONITRILE
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 14010 CHEMBL496879 PDB: U49 PubChem:23646577 PubChem:99445145 ZINC: ZINC000003870365
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.8 IC50 ChEMBL;BindingDB
P49356 FNTB Homo sapiens Human PF00432 8.8 IC50 ChEMBL
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P49354 FNTA Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha binder targets
P49356 FNTB Protein farnesyltransferase subunit beta binder targets