Molecule Details
InChIKeyUSLSTEHVCOVPEK-UHFFFAOYSA-N
Compound Name(2-Chloro-5-{4-[((2,4-difluorobenzyl){2-methyl-3-[(methylsulfonyl)amino]phenyl}amino)methyl]phenoxy}phenoxy)acetic acid
Canonical SMILESCc1c(NS(C)(=O)=O)cccc1N(Cc1ccc(Oc2ccc(Cl)c(OCC(=O)O)c2)cc1)Cc1ccc(F)cc1F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P04150 NR3C1 Homo sapiens Human PF02155 PF00104 PF00105 8.6 IC50 ChEMBL;BindingDB
P06401 PGR Homo sapiens Human PF00104 PF02161 PF00105 6.8 IC50 ChEMBL;BindingDB
P08235 NR3C2 Homo sapiens Human PF00104 PF00105 6.0 IC50 ChEMBL;BindingDB