Molecule Details
InChIKeyUSCKZBKHRWIQAC-UHFFFAOYSA-N
Compound NameN-(1-acetylpiperidin-4-yl)-5-(5-chloro-2,4-dihydroxyphenyl)-4-(4-methoxyphenyl)-1,2-oxazole-3-carboxamide
Canonical SMILESCOc1ccc(-c2c(C(=O)NC3CCN(C(C)=O)CC3)noc2-c2cc(Cl)c(O)cc2O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07900 HSP90AA1 Homo sapiens Human PF13589 PF00183 7.6 IC50 ChEMBL
P08238 HSP90AB1 Homo sapiens Human PF13589 PF00183 7.6 IC50 ChEMBL
Q15118 PDK1 Homo sapiens Human PF10436 PF02518 6.7 IC50 ChEMBL;BindingDB