Molecule Details
InChIKeyURTMWTKJLRDYRH-UHFFFAOYSA-N
Canonical SMILESCCN1C2CC1CN(c1ccc(Nc3ncc(F)c(-c4cc5c(=O)n(C)cc(C(C)C)c5s4)n3)nc1)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24385 CCND1 Homo sapiens Human PF02984 PF00134 7.0 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.0 IC50 ChEMBL