Molecule Details
InChIKeyURIHGJROOMIUNL-VWLOTQADSA-N
Canonical SMILESC[C@@]1(c2nc3cc(C(F)(F)F)ccc3[nH]2)CCCN1C(=O)c1cc(Br)ccc1-c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O43614 HCRTR2 Homo sapiens Human PF00001 PF03827 9.0 IC50 ChEMBL;BindingDB
O43613 HCRTR1 Homo sapiens Human PF00001 7.0 IC50 ChEMBL;BindingDB