Molecule Details
InChIKeyUQYCPGDIEUPDPU-UHFFFAOYSA-N
Compound Name4-[4-(Pyrrolidin-1-ylmethyl)piperidin-1-yl]thieno[3,2-d]pyrimidine-6-carboxamide
Canonical SMILESNC(=O)c1cc2ncnc(N3CCC(CN4CCCC4)CC3)c2s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.67
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NTG7 SIRT3 Homo sapiens Human PF02146 7.2 IC50 ChEMBL;BindingDB
Q8IXJ6 SIRT2 Homo sapiens Human PF02146 6.7 IC50 ChEMBL;BindingDB
Q96EB6 SIRT1 Homo sapiens Human PF02146 6.1 IC50 ChEMBL;BindingDB