Molecule Details
InChIKeyUQRQADYTKHCQGV-CSJROMOCSA-N
Compound Name(2S)-2-[[2-(2-methylphenyl)-4-[(E)-3-[(2-methylpropan-2-yl)oxy]-3-oxo-1-pyridin-3-ylprop-1-en-2-yl]benzoyl]amino]-4-methylsulfanylbutanoic acid
Canonical SMILESCSCC[C@H](NC(=O)c1ccc(/C(=C\c2cccnc2)C(=O)OC(C)(C)C)cc1-c1ccccc1C)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.82
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.8 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.8 IC50 ChEMBL