Molecule Details
InChIKeyUQKMSJFNACXHSL-HNNXBMFYSA-N
Compound Name2-[(2S)-1-[7-[(4,5-difluoro-1H-benzimidazol-2-yl)methylamino]-3-ethylpyrazolo[1,5-a]pyrimidin-5-yl]piperidin-2-yl]ethanol
Canonical SMILESCCc1cnn2c(NCc3nc4ccc(F)c(F)c4[nH]3)cc(N3CCCC[C@H]3CCO)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NYV4 CDK12 Homo sapiens Human PF00069 7.5 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.4 IC50 ChEMBL
P50750 CDK9 Homo sapiens Human PF00069 6.6 IC50 ChEMBL