Molecule Details
InChIKeyUQHCMUXJGZRDTC-ADYVUFBVSA-N
Compound NameH-Tyr-Cys(1)-Gly-D-Phe-D-Cys(1)-Arg-N(Me)Arg-Leu-NHEt
Canonical SMILESCCNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CCCN=C(N)N)N(C)C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H]1CSSC[C@H](NC(=O)[C@@H](N)Cc2ccc(O)cc2)C(=O)NCC(=O)N[C@H](Cc2ccccc2)C(=O)N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 10.2 IC50 ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB