Molecule Details
InChIKeyUPVAPSGKXAAHBG-CKTDUXNWSA-N
Canonical SMILESC[C@@H](O)[C@H](N)C(=O)NS(=O)(=O)OC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.31
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB03355
Drug Name5'-O-(L-Threonylsulfamoyl)adenosine
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 50366646 CHEMBL1163068 ChemSpider: 393081 PDB: TSB PubChem:445439 PubChem:46506859 ZINC: ZINC000015524571
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P26639 TARS1 Homo sapiens Human PF03129 PF02824 PF00587 PF07973 7.8 IC50 ChEMBL;BindingDB
Q8IIA4 Plasmodium falciparum (isolate 3D7) Pathogen PF03129 PF00587 PF07973 6.8 IC50 ChEMBL
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P0A8M5 P0A8M5 Threonine--tRNA ligase binder targets
Q8NW68 Q8NW68 Threonine--tRNA ligase binder targets